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Accelrys cdocker in discovery studio 2017 r2
Cdocker In Discovery Studio 2017 R2, supplied by Accelrys, used in various techniques. Bioz Stars score: 90/100, based on 1 PubMed citations. ZERO BIAS - scores, article reviews, protocol conditions and more
https://www.bioz.com/product/cdocker+in+discovery+studio+2017+r2/cdocker+in+discovery+studio+2017+r2/pm40199026-309-13-22
Average 90 stars, based on 1 article reviews
cdocker in discovery studio 2017 r2 - by Bioz Stars, 2026-10
90/100 stars

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Article Title: Discovery of 2,4-dianilinopyrimidine derivatives as novel p90 ribosomal S6 protein kinase (RSK) inhibitors.
Article Snippet: RSK, or p90 ribosomal S6 kinase, plays a crucial role in tumor cell proliferation and survival, making it an appealing target for cancer therapies.. With the aim to explore novel RSK inhibitors as anticancer agents, a series of 2,4-dianilinopyrimidine derivatives 2b–2n and 3a–3n have been designed and synthesized.. Among them, compound 3e displayed substantial kinase inhibitory activity against RSK2 (IC50 = 37.89 ± 3.08 nM) and a potent antiproliferative effect against a range of cell lines, including HeLa, MIA PaCa-2, U937, SW620, HT-29, AGS, and two kinds of EGFR mutant cells (IC50s = 0.189–0.572 μM).



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